SS-31

Also Known As: Elamipretide, MTP-131, Bendavia, SS-31 peptide, Szeto-Schiller 31, D-Arg-dimethylTyr-Lys-Phe-NH2, Cardiolipin-targeting peptide, Mitochondria-targeted peptide, Mitochondrial protective peptide, Inner mitochondrial membrane peptide, Cardiac mitochondria peptide, Bendavia heart failure, SS31 Barth syndrome, mitochondrial targeting, cardiolipin

SS-31 is a research-grade Mitochondria-targeted tetrapeptide targeting Cardiolipin on inner mitochondrial membrane studied in Anti-Aging & Longevity research. It is supplied strictly for in vitro laboratory research use only - not for human or animal consumption, and not FDA-approved.

Evidence Tier: Approved Drug - FDA and/or EMA approved with robust human trial data.

A mitochondria-protecting peptide newly approved for the rare Barth syndrome and studied broadly for mitochondrial and heart conditions.

At A Glance

SS-31 Key Research Facts
CategoryAnti-Aging & Longevity
Compound ClassMitochondria-targeted tetrapeptide (D-Arg-dimethylTyr-Lys-Phe-NH2); cardiolipin-targeting
Molecular TargetCardiolipin on inner mitochondrial membrane; scavenges mitochondrial ROS; stabilizes cristae architecture; restores respiratory chain efficiency
Molecular Weight639.79 Da
Amino Acid SequenceD-Arg-Dmt-Lys-Phe-NH2
CAS Number736992-21-5
Half-Life~4 hours
WADA Statusnot_listed
Evidence TierApproved Drug

Mechanism Of Action

It specifically binds to cardiolipin, a vital fat found on the inner wall of the mitochondria. This instantly restores the structural integrity of the cell's energy factory, improving ATP output.

Studied For

  • Primary mitochondrial disease
  • Barth syndrome (cardiolipin deficiency)
  • Heart failure / ischemia-reperfusion injury
  • Dry AMD (age-related macular degeneration)
  • Mitochondrial aging
  • Cardiac energetics
  • Skeletal muscle mitochondria
  • Kidney ischemia-reperfusion models
  • ROS reduction at mitochondria
  • Cardiolipin stabilization
  • Respiratory chain Complex I-V efficiency
  • ATP production enhancement
  • Frailty / aging mitochondria
  • Chronic kidney disease models
  • Neurodegenerative disease mitochondria
  • Exercise intolerance research
  • energy production
  • anti-aging
  • mitochondrial repair
  • heart failure
  • cognitive decline
  • ischemia reperfusion
  • kidney protection

Reported Research Findings

The Barth-syndrome trial (TAZPOWER) supported a 2025 FDA accelerated approval for Barth syndrome; the primary mitochondrial myopathy program (MMPOWER-3) failed its endpoints, and several cardiac and dry-AMD endpoints were mixed or not met. Still the strongest human evidence in this group.

Safety And Handling Notes

Injection-site reactions, headache, gastrointestinal symptoms; generally tolerable at studied doses.

The 2025 accelerated approval is narrow (Barth syndrome, patients at least 30 kg); accelerated approval is conditional on confirmatory evidence. All other uses remain investigational and several large trials did not meet their endpoints. Research use only outside approved labeling.

Regulatory Status

FDA accelerated approval 19 September 2025 as Forzinity (elamipretide hydrochloride) to improve muscle strength in adult and pediatric patients with Barth syndrome weighing at least 30 kg; 40 mg subcutaneous once daily. Holds FDA Orphan Drug, Fast Track, Priority Review and Rare Pediatric designations, and an EMA Orphan Drug designation for Barth syndrome. No EMA marketing authorization identified as of August 2026. All other uses remain investigational. Not on the WADA 2026 Prohibited List.

Full Reference Detail

Related Research Guides

Maintained By The Pep Nation Lab Research Team. See Our Editorial Standards And Research Methodology For How This Reference Is Sourced And Reviewed.

This Reference Is Provided For In Vitro Laboratory Research Use Only. Not For Human Consumption. See The Full Research Disclaimer.

References And Citations

  1. PubMed / NCBI Reference
  2. neurology.org
  3. nature.com
Spec Sheet

SS-31

Also Known As: Elamipretide, MTP-131, Bendavia, SS-31 peptide, Szeto-Schiller 31, D-Arg-dimethylTyr-Lys-Phe-NH2, Cardiolipin-targeting peptide, Mitochondria-targeted peptide, Mitochondrial protective peptide, Inner mitochondrial membrane peptide, Cardiac mitochondria peptide, Bendavia heart failure, SS31 Barth syndrome, mitochondrial targeting, cardiolipin

Approved DrugAnti-Aging & Longevity

Explain Like I'm 5

  • SS-31 acts like a mechanic that specifically repairs the engine inside your cells (the mitochondria). By fixing the engines, it brings dead, tired cells back to life, reversing aging at the deepest possible level.

A mitochondria-protecting peptide newly approved for the rare Barth syndrome and studied broadly for mitochondrial and heart conditions.

Identity & Classification
SS-31 Key Research Facts
ClassMitochondria-targeted tetrapeptide (D-Arg-dimethylTyr-Lys-Phe-NH2); cardiolipin-targeting
Molecular TargetCardiolipin on inner mitochondrial membrane; scavenges mitochondrial ROS; stabilizes cristae architecture; restores respiratory chain efficiency
CategoryAnti-Aging & Longevity
Molecular Weight639.79 Da
Amino Acid SequenceD-Arg-Dmt-Lys-Phe-NH2
CAS Number736992-21-5
Parent CompoundSzeto-Schiller peptide series
Research Metrics at a Glance
473
PubMed Citations

Related Compounds

Research Use Only. Not For Human Or Veterinary Use. Information Provided For Laboratory Research Purposes Only.

Research Reference Only — Not Medical Advice. For In Vitro Laboratory Use Only.
Typical Dose2–4 mg/kg (rodent models); typical human-equivalent: 0.05–0.25 mg/kg
FrequencyOnce daily (or infusion in some cardiac research protocols)
Cycle On4–8 weeks
Cycle Off4 weeks
Route(s)
SubcutaneousIntravenous (research infusion)
Research Notes

Mitochondria-targeted antioxidant peptide (Szeto-Schiller peptide). Most cardiac and mitochondrial research uses IV infusion at controlled rates. Subcutaneous used for chronic dosing research. Human-equivalent doses derived from allometric scaling of published rodent data.

Sequence Motif Viewer

21 Residues
D-ARG-DMT-LYS-PHE-NH2
BasicAcidicPolarNon-PolarAromaticSpecial
CompoundCompoundTargetReceptor / TargetIt specifically bind...Downstream PathwayResearch EffectStudied Effect

Compare SS-31

SS-31 Frequently Asked Questions

What Is SS-31?

A mitochondria-protecting peptide newly approved for the rare Barth syndrome and studied broadly for mitochondrial and heart conditions.

How Does SS-31 Work?

It specifically binds to cardiolipin, a vital fat found on the inner wall of the mitochondria. This instantly restores the structural integrity of the cell's energy factory, improving ATP output.

What Has SS-31 Been Studied For?

In the referenced literature, SS-31 has been studied for Primary mitochondrial disease, Barth syndrome (cardiolipin deficiency), Heart failure / ischemia-reperfusion injury, Dry AMD (age-related macular degeneration), Mitochondrial aging, Cardiac energetics, Skeletal muscle mitochondria, Kidney ischemia-reperfusion models, ROS reduction at mitochondria, Cardiolipin stabilization, Respiratory chain Complex I-V efficiency, ATP production enhancement, Frailty / aging mitochondria, Chronic kidney disease models, Neurodegenerative disease mitochondria, Exercise intolerance research, energy production, anti-aging, mitochondrial repair, heart failure, cognitive decline, ischemia reperfusion, kidney protection. This summarizes research focus only and is not a claim of efficacy.

What Is The Reported Half-Life Of SS-31?

SS-31 has a reported half-life of ~4 hours in the referenced literature.

Is SS-31 Approved For Human Use?

No. SS-31 is supplied strictly for in vitro laboratory research use only. It is not intended for human or animal consumption, ingestion, or injection, and it has not been evaluated by the FDA.

Regional Research Availability

Pep Nation Lab supplies research-grade SS-31 to qualified researchers and scientific institutions nationwide. Browse verified availability and per-region documentation by state:

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