MT-1

Also Known As: Afamelanotide, Scenesse, NDP-MSH, Melanotan I, Melanotan 1, MT1, [Nle4-D-Phe7]-alpha-MSH, Norleucine 4 D-phenylalanine 7 alpha-MSH analog, Photoprotective peptide, Tanning peptide, EPP treatment peptide, MC1R agonist peptide, Melanocortin 1 agonist, tanning peptide

MT-1 is a research-grade Synthetic alpha-MSH analog with [Nle4 targeting MC1R studied in Skin, Hair & Cosmetics research. It is supplied strictly for in vitro laboratory research use only - not for human or animal consumption, and not FDA-approved.

Evidence Tier: Approved Drug - FDA and/or EMA approved with robust human trial data.

An approved melanocortin drug for a rare light-sensitivity disease; needs skin monitoring.

At A Glance

MT-1 Key Research Facts
CategorySkin, Hair & Cosmetics
Compound ClassSynthetic alpha-MSH analog with [Nle4,D-Phe7] substitutions; MC1R-selective agonist
Molecular TargetMC1R (melanocortin-1 receptor) on melanocytes; stimulates eumelanin synthesis and photoprotection
Molecular Weight1646.86 Da
Amino Acid SequenceAc-Ser-Tyr-Ser-Nle-Glu-His-D-Phe-Arg-Trp-Gly-Lys-Pro-Val-NH2
CAS Number75921-69-6
Half-Life~30 minutes
WADA Statusnot_listed
Evidence TierApproved Drug

Mechanism Of Action

It binds to the melanocortin 1 receptor on skin cells, stimulating the production of melanin (the dark pigment) while remaining very safe and not crossing into the brain to cause side effects.

Studied For

  • Erythropoietic protoporphyria (EPP) (FDA/EMA approved)
  • Photodermatoses research
  • Solar urticaria
  • Polymorphous light eruption (PLE)
  • UV light protection
  • Melanin production stimulation
  • Skin darkening / tanning research
  • Squamous cell carcinoma prevention research
  • Libido research (MC4R pathway)
  • Melanocortin system research
  • Vitiligo models
  • Inflammatory skin disease models
  • skin pigmentation
  • sunless tan
  • phototoxicity prevention
  • vitiligo
  • erythropoietic protoporphyria

Reported Research Findings

Phase 3 trials in erythropoietic protoporphyria showed increased pain-free sun exposure, the basis for FDA and EMA approval as a controlled-release implant.

Safety And Handling Notes

Implant-site reactions, headache, nausea, and darkening of moles, which warrants periodic skin monitoring.

An approved orphan drug delivered as a physician-administered implant; distinct from unregulated melanotan products. Requires skin-lesion surveillance.

Regulatory Status

FDA (2019) and EMA (2014) approved for EPP.

Full Reference Detail

Related Research Guides

Maintained By The Pep Nation Lab Research Team. See Our Editorial Standards And Research Methodology For How This Reference Is Sourced And Reviewed.

This Reference Is Provided For In Vitro Laboratory Research Use Only. Not For Human Consumption. See The Full Research Disclaimer.

References And Citations

  1. go.drugbank.com
  2. ema.europa.eu
Spec Sheet

MT-1

Also Known As: Afamelanotide, Scenesse, NDP-MSH, Melanotan I, Melanotan 1, MT1, [Nle4-D-Phe7]-alpha-MSH, Norleucine 4 D-phenylalanine 7 alpha-MSH analog, Photoprotective peptide, Tanning peptide, EPP treatment peptide, MC1R agonist peptide, Melanocortin 1 agonist, tanning peptide

Approved DrugSkin, Hair & Cosmetics

Explain Like I'm 5

  • Melanotan-1 mimics a natural hormone that tells your skin to produce a protective, dark tan without needing to sit in the sun for hours. It provides a flawless tan while protecting the skin from UV damage.

An approved melanocortin drug for a rare light-sensitivity disease; needs skin monitoring.

Identity & Classification
MT-1 Key Research Facts
ClassSynthetic alpha-MSH analog with [Nle4,D-Phe7] substitutions; MC1R-selective agonist
Molecular TargetMC1R (melanocortin-1 receptor) on melanocytes; stimulates eumelanin synthesis and photoprotection
CategorySkin, Hair & Cosmetics
Molecular Weight1646.86 Da
Amino Acid SequenceAc-Ser-Tyr-Ser-Nle-Glu-His-D-Phe-Arg-Trp-Gly-Lys-Pro-Val-NH2
CAS Number75921-69-6
Parent Compoundalpha-MSH analog
Research Metrics at a Glance
1,940
PubMed Citations
5
Clinical Trials
5 Active

Related Compounds

Research Use Only. Not For Human Or Veterinary Use. Information Provided For Laboratory Research Purposes Only.

Research Reference Only — Not Medical Advice. For In Vitro Laboratory Use Only.
Typical Dose0.5–1 mg
FrequencyOnce daily (loading); 2–3 times/week (maintenance)
Cycle On2–4 weeks loading; ongoing maintenance
Cycle OffTanning effect fades over 4–8 weeks post-cycle
Route(s)
Subcutaneous
Research Notes

Melanotan I (afamelanotide). Linear ACTH/MSH analogue. FDA approved as Scenesse for erythropoietic protoporphyria. Research tanning protocols start at 0.5 mg to assess tolerance. Nausea common at higher doses. Melanocytes activated over 2–4 week period.

Sequence Motif Viewer

60 Residues
AC-SER-TYR-SER-NLE-GLU-HIS-D-PHE-ARG-TRP-GLY-LYS-PRO-VAL-NH2
BasicAcidicPolarNon-PolarAromaticSpecial
CompoundCompoundTargetReceptor / TargetIt binds to the mela...Downstream PathwayResearch EffectStudied Effect

MT-1 Frequently Asked Questions

What Is MT-1?

An approved melanocortin drug for a rare light-sensitivity disease; needs skin monitoring.

How Does MT-1 Work?

It binds to the melanocortin 1 receptor on skin cells, stimulating the production of melanin (the dark pigment) while remaining very safe and not crossing into the brain to cause side effects.

What Has MT-1 Been Studied For?

In the referenced literature, MT-1 has been studied for Erythropoietic protoporphyria (EPP) (FDA/EMA approved), Photodermatoses research, Solar urticaria, Polymorphous light eruption (PLE), UV light protection, Melanin production stimulation, Skin darkening / tanning research, Squamous cell carcinoma prevention research, Libido research (MC4R pathway), Melanocortin system research, Vitiligo models, Inflammatory skin disease models, skin pigmentation, sunless tan, phototoxicity prevention, vitiligo, erythropoietic protoporphyria. This summarizes research focus only and is not a claim of efficacy.

What Is The Reported Half-Life Of MT-1?

MT-1 has a reported half-life of ~30 minutes in the referenced literature.

Is MT-1 Approved For Human Use?

No. MT-1 is supplied strictly for in vitro laboratory research use only. It is not intended for human or animal consumption, ingestion, or injection, and it has not been evaluated by the FDA.

Regional Research Availability

Pep Nation Lab supplies research-grade MT-1 to qualified researchers and scientific institutions nationwide. Browse verified availability and per-region documentation by state:

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