The Appetite Crusher Stack

Also Known As: CagriSema, CagriSema combination, Cagrilintide semaglutide, AM833 NN9535, Amylin GLP-1 dual agonist, Dual obesity drug, CagriSema stack, Amylin analog + GLP-1 agonist, Anti-obesity dual therapy, CagriSema combo, Cagrilintide with semaglutide, cagrilintide + semaglutide

The Appetite Crusher Stack is a research-grade Fixed-ratio combination: long-acting amylin analog targeting Amylin/calcitonin receptors studied in Weight Loss & Metabolism research. It is supplied strictly for in vitro laboratory research use only - not for human or animal consumption, and not FDA-approved.

Evidence Tier: Investigational - In active human clinical trials; not yet approved.

An investigational amylin-plus-GLP-1 combination with strong trial weight loss.

At A Glance

The Appetite Crusher Stack Key Research Facts
CategoryWeight Loss & Metabolism
Compound ClassFixed-ratio combination: long-acting amylin analog (cagrilintide) + GLP-1 receptor agonist (semaglutide)
Molecular TargetAmylin/calcitonin receptors (cagrilintide) + GLP-1 receptor (semaglutide); dual satiety and glucose regulation
Molecular Weightcombination
Amino Acid Sequencecagrilintide + semaglutide
CAS Numbern/a
Half-Life~1 week (both components weekly SC)
WADA Statusnot_listed
Evidence TierInvestigational

Mechanism Of Action

It hits the brain from two different angles. It activates the GLP-1 switch (which controls blood sugar and cravings) and the Amylin switch (which controls physical fullness in the stomach).

Studied For

  • Obesity / overweight
  • Type 2 diabetes
  • Dual-mechanism weight loss
  • GLP-1 plus amylin dual therapy
  • Cardiometabolic disease
  • HbA1c reduction
  • Appetite suppression dual pathway
  • Body weight reduction
  • Metabolic syndrome
  • Insulin resistance
  • Blood sugar control
  • Caloric intake reduction research
  • Combination incretin amylin therapy
  • Cardiovascular risk reduction
  • obesity
  • appetite suppression
  • extreme weight loss
  • metabolic control

Reported Research Findings

Phase 3 REDEFINE 1 (2025, 68 weeks) reported about 22.7 percent mean body-weight reduction in obesity, exceeding either component alone.

Safety And Handling Notes

Predominantly gastrointestinal, consistent with both component classes.

Investigational with no approved indication. Inherits the GLP-1 class thyroid C-cell and pancreatitis considerations. Research use only.

Regulatory Status

Investigational (Novo Nordisk); NDA filed with FDA 18 Dec 2025 on the REDEFINE 1 and REDEFINE 2 pivotal trials and under FDA review through 2026; company guidance points to a decision in Q4 2026, and no PDUFA date has been publicly confirmed. Would be the first once-weekly GLP-1 plus amylin analogue combination for weight management if approved. Note that the Phase 3 REDEFINE 4 head-to-head trial did not meet its primary endpoint of non-inferiority on weight loss versus tirzepatide at 84 weeks. Not approved.

Full Reference Detail

Related Research Guides

Maintained By The Pep Nation Lab Research Team. See Our Editorial Standards And Research Methodology For How This Reference Is Sourced And Reviewed.

This Reference Is Provided For In Vitro Laboratory Research Use Only. Not For Human Consumption. See The Full Research Disclaimer.

References And Citations

  1. en.wikipedia.org
Spec Sheet

The Appetite Crusher Stack

Also Known As: CagriSema, CagriSema combination, Cagrilintide semaglutide, AM833 NN9535, Amylin GLP-1 dual agonist, Dual obesity drug, CagriSema stack, Amylin analog + GLP-1 agonist, Anti-obesity dual therapy, CagriSema combo, Cagrilintide with semaglutide, cagrilintide + semaglutide

InvestigationalWeight Loss & MetabolismGLP-1 Class

Explain Like I'm 5

  • CagriSema is a super-team of two weight-loss signals. One tells your stomach to stay full, and the other tells your brain to stop craving sugar. Working together, they cause massive weight loss without feeling starved.

An investigational amylin-plus-GLP-1 combination with strong trial weight loss.

Identity & Classification
The Appetite Crusher Stack Key Research Facts
ClassFixed-ratio combination: long-acting amylin analog (cagrilintide) + GLP-1 receptor agonist (semaglutide)
Molecular TargetAmylin/calcitonin receptors (cagrilintide) + GLP-1 receptor (semaglutide); dual satiety and glucose regulation
CategoryWeight Loss & Metabolism
Molecular Weightcombination
Amino Acid Sequencecagrilintide + semaglutide
CAS Numbern/a
Parent CompoundCagrilintide and Semaglutide
Classification Flags
GLP-1 / Incretin Class
Stack Components
cagrilintidesemaglutide

Related Compounds

Research Use Only. Not For Human Or Veterinary Use. Information Provided For Laboratory Research Purposes Only.

Research Reference Only — Not Medical Advice. For In Vitro Laboratory Use Only.
Typical DoseCagrilintide 2.4 mg + Semaglutide 2.4 mg (co-formulated)
FrequencyOnce weekly
Cycle On68+ weeks (per REDEFINE Phase 3 trial)
Cycle OffNot yet established
Route(s)
Subcutaneous
Research Notes

Fixed-ratio combination of cagrilintide + semaglutide under investigation by Novo Nordisk. Phase 2 data (2022) showed up to 15.6% weight loss at 32 weeks. Phase 3 REDEFINE program ongoing. Dose-limiting nausea/vomiting addressed via slow titration.

Sequence Motif Viewer

24 Residues
CAGRILINTIDE+SEMAGLUTIDE
BasicAcidicPolarNon-PolarAromaticSpecial
CompoundCompoundTargetReceptor / TargetIt hits the brain fr...Downstream PathwayResearch EffectStudied Effect

Compare The Appetite Crusher Stack

The Appetite Crusher Stack Frequently Asked Questions

What Is The Appetite Crusher Stack?

An investigational amylin-plus-GLP-1 combination with strong trial weight loss.

How Does The Appetite Crusher Stack Work?

It hits the brain from two different angles. It activates the GLP-1 switch (which controls blood sugar and cravings) and the Amylin switch (which controls physical fullness in the stomach).

What Has The Appetite Crusher Stack Been Studied For?

In the referenced literature, The Appetite Crusher Stack has been studied for Obesity / overweight, Type 2 diabetes, Dual-mechanism weight loss, GLP-1 plus amylin dual therapy, Cardiometabolic disease, HbA1c reduction, Appetite suppression dual pathway, Body weight reduction, Metabolic syndrome, Insulin resistance, Blood sugar control, Caloric intake reduction research, Combination incretin amylin therapy, Cardiovascular risk reduction, obesity, appetite suppression, extreme weight loss, metabolic control. This summarizes research focus only and is not a claim of efficacy.

What Is The Reported Half-Life Of The Appetite Crusher Stack?

The Appetite Crusher Stack has a reported half-life of ~1 week (both components weekly SC) in the referenced literature.

Is The Appetite Crusher Stack Approved For Human Use?

No. The Appetite Crusher Stack is supplied strictly for in vitro laboratory research use only. It is not intended for human or animal consumption, ingestion, or injection, and it has not been evaluated by the FDA.

Regional Research Availability

Pep Nation Lab supplies research-grade The Appetite Crusher Stack to qualified researchers and scientific institutions nationwide. Browse verified availability and per-region documentation by state:

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